Tranexamic acid

Generic Name: Tranexamic

Brand Names:

Availability: Available with Prescription

Drug Class: Antifibrinolytics

Therapeutic action

  • Antifibrinolytic

Indications

  • Abnormal uterine bleeding (especially functional uterine bleeding unrelated to pregnancy)

Forms and strengths

  • 500 mg tablet

Dosage and duration

  • Adolescent and adult: 1 g 3 times daily (max. 1 g 4 times daily) until bleeding stops (max. 5 days)

Contra-indications, adverse effects, precautions

  • Do not administer in patients with (or with history of) venous or arterial thromboembolic disorders, severe renal impairment, history of seizures.
  • Reduce dosage in patients with mild to moderate renal impairment (risk of accumulation).
  • May cause: gastrointestinal disturbances, seizures with high doses, visual disturbances, allergic reactions.
  • Avoid combination with drugs that increase the risk of thromboembolism. Concomitant use of oestrogens (e.g. ethinylestradiol/levonorgestrel) should be carefully considered on a case-by-case basis.
  • Pregnancy: this drug is not indicated in the event of bleeding during pregnancy.
  • Breast-feeding: no contra-indication

Remarks

  • The treatment may be administered at each bleeding episode. In situations of repeated bleeding,it may be helpful to combine tranexamic acid with a non-steroidal anti-inflammatory drug and/or a long-term treatment with a levonorgestrel intrauterine device or ethinylestradiol/levonorgestrel or oral or injectable medroxy progesterone.

Storage

- Below 25 °C